Description
Our GW501516 Cardarine liquid comes as 30mL of ready-made solution at 10mg/mL, so each bottle holds 300mg of GW501516 (cardarine), a PPAR-delta agonist. This batch tested at 99.34% purity. It’s sold for laboratory research only.
GW501516 (cardarine) at a glance
GW501516 (cardarine) is a PPAR-delta agonist developed by GlaxoSmithKline and Ligand in the 1990s. It’s often sold next to SARMs, but it works through a different receptor, one that switches on fat-burning genes in muscle.
GSK stopped development after rodent studies linked long-term high exposure to cancer in several organs. It’s on the WADA prohibited list.
GW501516 mechanism of action
PPAR-delta is a nuclear receptor. When GW501516 binds it, it pairs with the retinoid X receptor and switches on genes for taking up and burning fatty acids, such as CPT1 and PDK4.
In muscle, that shifts fuel use from glucose toward fat and pushes fibers toward the slow-twitch, fatigue-resistant type. That’s the basis for the endurance results in mice.
GW501516 Cardarine liquid specifications
- Compound: GW501516 (cardarine)
- Also known as: cardarine, GW-501516, endurobol
- CAS number: 317318-70-0
- Molecular formula: C21H18F3NO3S2
- Molar mass: 453.5 g/mol
- Structure: phenoxyacetic acid with a thiazole ring
- Concentration: 10mg/mL
- Volume: 30mL (300mg in total)
- Form: ready-made liquid in a glass dropper bottle
- Purity: 99.34% (mass spectrometry and HPLC-UV)
- SKU: BSP-GW-30
- Use: laboratory research only
What the research says about GW501516
Narkar and colleagues showed in Cell in 2008 that GW501516 combined with exercise or with AICAR raised running endurance in mice and shifted muscle toward slow-twitch fibers.
Earlier work by Oliver and colleagues, published in PNAS in 2001, reported higher HDL cholesterol and lower triglycerides in obese rhesus monkeys.
To read the papers yourself, start with this PubMed search for GW501516.
How GW501516 compares
Here’s how GW501516 Cardarine liquid fits among related compounds. GW501516 is a PPAR-delta agonist that shifts muscle toward burning fat, not a SARM. By comparison:
- MK-2866 is the most studied SARM, with a phase 2 trial in cancer-related muscle loss
- LGD-4033 binds the androgen receptor very tightly and has a published phase 1 study
- RAD-140 showed strong muscle selectivity in monkeys and was trialed in breast cancer
- S4 Andarine is a partial androgen receptor agonist, one of the first SARMs from GTx
- YK-11 is a steroidal partial agonist that raises follistatin in muscle cells
- MK-677 is an oral ghrelin mimic that raises GH and IGF-1, not a SARM
Only the first five act on the androgen receptor. MK-677 and GW501516 are sold alongside SARMs because they’re studied for body composition too, but they work through different receptors. See them all on our SARMs page.
Working with GW501516 Cardarine liquid
The concentration is 10mg/mL, so the math is simple: every 1mL holds 10mg, and every 0.1mL holds 1mg. The whole 30mL bottle holds 300mg.
Most labs measure with a 1mL measuring dropper marked in 0.1mL steps. The dropper built into the cap is handy for transfers but not precise enough for measuring.
GW501516 Cardarine liquid storage and shelf life
Keep GW501516 Cardarine liquid at room temperature with the cap tight, out of direct sunlight. It doesn’t need a fridge. Wipe the dropper tip before you put the cap back so nothing dries in the threads.
Lab-tested GW501516 Cardarine liquid
Our GW501516 Cardarine liquid batch measured 99.34% pure by HPLC with mass spectrometry confirming the identity. We print the real number, so you know what’s going into your experiment.
The label on each bottle shows the compound, the strength and the batch. Ask us for the certificate of analysis for your batch and we’ll email it over.
If a result looks off, check the batch number first, then your handling notes. Most problems with GW501516 come from storage or mixing, not the material.
Compounds often ordered with GW501516
- MK-2866 Ostarine Liquid 35mg/mL (30mL), a SARM in a 30mL bottle
- LGD-4033 Liquid 10mg/mL (30mL), a SARM in a 30mL bottle
- YK-11 Liquid 10mg/mL (30mL), a steroidal SARM in a 30mL bottle
- RAD-140 Liquid 10mg/mL (30mL), a SARM in a 30mL bottle
- S4 Andarine Liquid 25mg/mL (30mL), a SARM in a 30mL bottle
Browse the full SARMs range, or see everything on our research liquids page.
Common questions about GW501516 Cardarine liquid
How much is in the GW501516 Cardarine liquid bottle?
30mL of solution at 10mg/mL, which is 300mg in total. The amount is printed on the label.
Can GW501516 be used in people or animals?
No. It’s sold for laboratory research only and isn’t approved for human or veterinary use.
Is GW501516 Cardarine liquid in stock?
Yes, GW501516 Cardarine liquid is in stock now and ready to ship.
Is there a COA for GW501516 Cardarine liquid?
Yes. Each batch has a certificate of analysis filed under the batch number on the label. Email us that number and we’ll send it.
Does GW501516 Cardarine liquid need mixing?
No. It’s already a solution in a dropper bottle, so there’s no powder to reconstitute.
Buy GW501516 Cardarine liquid online
Ready to order? GW501516 Cardarine liquid costs $63.67 and is in stock. Add it to your cart and you’re done.
Need more for the same project? See the rest of our SARMs.
For laboratory research use only. Not for human or veterinary use. Not evaluated by the FDA.
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